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Michango
Majadiliano
Kigezo
:
GABAergics
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Ongeza viungo
Kigezo
Majadiliano
Kiswahili
Soma
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Zana
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Ukurasa wa kuchapika
Kutoka Wikipedia, kamusi elezo huru
v
d
e
GABAergics
Receptor
ligands
GABA
A
Agonists:
Main site:
Bamaluzole
•
Gaboxadol
•
Ibotenic acid
•
Isoguvacine
•
Isonipecotic acid
•
Muscimol
(
Amanita Muscaria
) •
Progabide
•
SL 75102
•
Thiomuscimol
•
Tolgabide
;
Positive allosteric modulators
:
Barbiturates
•
Benzodiazepines
•
Carbamates
•
Chlormezanone
•
Clomethiazole
•
Ethanoli
(Alcohol) •
Etomidate
•
Kavalactones
(
Kava kava
) •
Loreclezole
•
Neuroactive steroids
•
Nonbenzodiazepines
•
Phenols
•
Piperidinediones
•
Propanidid
•
Pyrazolopyridines
•
Quinazolinones
•
ROD-188
•
Skullcap
•
Stiripentol
•
Thymol
•
Valerenic acid
(
Valerian
)
* See
Template:GABAAergics
for a full list of GABA
A
positive allosteric modulators.
Antagonists:
Main site:
Bicuculline
•
Gabazine
•
Pitrazepin
;
Negative allosteric modulators
:
α5IA
•
Bilobalide
•
Cicutoxin
•
Cyclothiazide
•
DMCM
•
Flumazenil
•
Flurothyl
•
Furosemide
•
L-655,708
•
Oenanthotoxin
•
Penicillin
•
Pentylenetetrazol
•
Picrotoxin
•
PWZ-029
•
Ro15-4513
•
Sarmazenil
•
Suritozole
•
Thujone
(
Absinthe
) •
Thiocolchicoside
GABA
B
Agonists:
Main site:
1,4-Butanediol
•
Baclofen
•
GBL
•
GHB
•
GHV
•
GVL
•
Lesogaberan
•
Phenibut
•
Progabide
•
SKF-97,541
•
Tolgabide
;
Positive allosteric modulators
:
BHF-177
•
BHFF
•
BSPP
•
CGP-7930
•
GS-39783
Antagonists:
Main site:
CGP-35348
•
Phaclofen
•
Saclofen
•
SCH-50911
GABA
C
Agonists:
Main site:
CACA
•
CAMP
•
GABOB
•
N(4)-chloroacetylcytosine arabinoside
•
Progabide
•
Tolgabide
Antagonists:
Main site:
Bilobalide
•
TPMPA
Reuptake
inhibitors
Plasmalemmal
GAT
inhibitors
CI-966
•
Deramciclane
•
EF-1502
•
Gabaculine
•
Guvacine
•
Nipecotic acid
•
NNC 05-2090
•
SKF-89976A
•
SNAP-5114
•
Tiagabine
Enzyme
inhibitors
Anabolism
GAD
inhibitors
Allylglycine
Catabolism
GABA-T
inhibitors
3-Hydrazinopropionic acid
•
Aminooxyacetic acid
•
Gabaculine
•
Isoniazid
•
Phenelzine
•
Phenylethylidenehydrazine
•
Sodium valproate
•
Valnoctamide
•
Valproate pivoxil
•
Valproate semisodium
(Divalproex sodium) •
Valproic acid
•
Valpromide
•
Vigabatrin
Others
Precursors
Glutamate
•
Glutamine
Cofactors
Vitamin B6
(
pyridoxine
,
pyridoxamine
,
pyridoxal phosphate
)
Others
Gabapentin
•
L-Theanine
•
Picamilon
•
Pregabalin
Jamii
:
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